77-301-0
Tocris Bioscience™ AS2717638
Manufacturer: Tocris Bioscience™
CAS Number: 2148339-28-8
Select a Size
| Pack Size | SKU | Availability | Price |
|---|---|---|---|
| Each of 1 | 77-301-0-Each-of-1 | In Stock | ₹ 27,323.00 |
77-301-0 - Each of 1
In Stock
Quantity
1
Base Price: ₹ 27,323.00
GST (18%): ₹ 4,918.14
Total Price: ₹ 32,241.14
Chemical Name or Material
6,7-Dimethoxy-2-(5-methyl-1,2-benzisoxazol-3-yl)-4-(1-piperidinylcarbonyl)-1(2 H)-isoquinolinone
Quantity
10 mg
Molecular Formula
C25H25N3O5
CAS
2148339-28-8
Target
LPAR5/LPA5/GPR92
Purity
0.98
Other Options
| Image | Product Name | Manufacturer | Price Range | |
|---|---|---|---|---|
Medchemexpress LLC HY-114379 5mg Medchemexpress, AS2717638 CAS:2148339-28-8 Purity:>98% | -- | ₹ 36,445.50 | ||
2148339-28-8 | AS2717638 | -- | ₹ 5,785.00 - ₹ 99,324.00 |
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Description
- AS2717638 is a potent LPA5 receptor antagonist (IC50 = 38 nM in BV-2 microglia cells)
- It is selective for LPA5 over LPA1, LPA2, and LPA3
- It inhibits LPA-mediated pro-inflammatory transcription factor phosphorylation
- In vivo , AS2717638 inhibits LPA5 agonist-induced allodynia in mice
- It also exhibits analgesic effects against both neuropathic and inflammatory pain in rodent models
- Orally bioavailable and brain penetrant.
SAFETY INFORMATION
- Recommended Storage : Store at -20°C