7112433

Tocris Bioscience™ TASP 0390325

Potent and selective V1B receptor antagonist; orally bioavailable

Manufacturer: Fischer Scientific

CAS Number: 1642187-96-9

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Product Type

Antagonist

CAS

1642187-96-9

Formula Weight

554.44g/mol

For Use With (Application)

Vasopressin Receptor Antagonists

Target Proteins

Vasopressin Receptor

Molecular Formula

C25H29ClFN5O4.HCl

Content And Storage

Store at -20°C

Other Options

Image Product Name Manufacturer Price Range
Tocris Bioscience™ TASP 0390325
-- ₹ 29,014.00
Tocris Bioscience™ TASP 0390325
-- ₹ 1,20,506.00
1642187-96-9 | 2-(2-(3-Chloro-4-fluorophenyl)-6-(3-morpholinopropoxy)-4-oxopyrido[2,3-d]pyrimidin-3(4H)-yl)-N-isopropylacetamide hydroChloride
-- ₹ 17,177.00 - ₹ 1,48,007.00

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Description

  • Potent and selective V1B receptor antagonist (IC50 = 2.22 nM for rat pituitary receptor)
  • Exhibits no significant affinity for 85 other receptors, ion channels and transporters at 10 μM, including V1A and V2
  • Increases ACTH levels in rats
  • Orally bioavailable
  • Antidepressant and anxiolytic.